P53 Tumor Suppressor Protein Activating

The invention provides a compound of formula (I), wherein X, L1-4 and R1-4 are as defined herein, with the proviso that the compound is not (i) 4-benzoyl-3,5-dimethyl-1H-pyrrole-2-carboxylic acid ethyl ester; (ii) 4-(2,5-difluorobenzoyl)-3,5-dimethyl-1H-pyrrole-2-carboxylic acid ethyl ester); (iii) 4-acetyl-3,5-dimethyl-1H-pyrrole-2-carboxylic acid ethyl ester; or (iv) 4-(3-dimethylamino-acryloyl)-3,5-dimethyl-1H-pyrrole-2-carboxylic acid ethyl ester, or a pharmaceutically acceptable derivative thereof.

Attached files:


Patents:
WO 2,010,013,011

Inventor(s): WESTWOOD NICHOLAS JAMES [GB]; LAIN SONIA [SE]; HOLLICK JONATHAN JAMES [GB]; LANE DAVID PHILIP [GB]

Type of Offer: Sale



« More Pharmaceutical Patents

---