Unique Dual-action Therapeutics

A new family of therapeutics which provides a controlled-release delivery platform for non-steroidal anti-inflammatory agents on an ester or an ester-carbonate backbone is disclosed herein. These agents are reversible inhibitors of acetylcholinesterase and are thus useful for clinical conditions benefiting from inflammation suppression and cholinergic intervention. These compounds are of the general formula wherein n = 0, 1; X = C, Si, and N+ and NSAID = ibuprofen, naproxen, indomethacin and diclofenac. Other embodiments are also disclosed.

Attached files:


Patents:
WO 2,010,051,044

Inventor(s): LASKIN JEFFREY [US]; HECK DIANE [US]; HUAN MOU-TUAN [US]; FABIO KARINE [US]; LACEY C JEFFREY; YOUNG SHERRI [US]; MOHANTA PRAMOD

Type of Offer: Licensing



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